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SOURCE:
Experimental database
Expanded database
PROPERTY:
None
None
【Basic】LogD7.4
【Basic】LogP
【Basic】LogS
【Absorption】Caco-2
【Absorption】Pgp-inhibitor
【Absorption】Pgp-substrate
【Absorption】F (30%)
【Distribution】PPB
【Distribution】BBB
【Distribution】vdss
【Metabolism】CYP 1A2-inhibitor
【Metabolism】CYP 2C19-inhibitor
【Metabolism】CYP 2C9-inhibitor
【Metabolism】CYP 2D6-inhibitor
【Metabolism】CYP 2d6-substrate
【Metabolism】CYP 3A4-inhibitor
【Excretion】T
1/2
【Toxicity】Ames
【Toxicity】BCF
【Toxicity】DILI
【Toxicity】EC
【Toxicity】EI
【Toxicity】FDAMDD
【Toxicity】H-HT-2
【Toxicity】hERG
【Toxicity】IGC50
【Toxicity】NR-AhR
【Toxicity】NR-AR
【Toxicity】NR-AR-LBD
【Toxicity】Respiratory
【Toxicity】SR-ARE
【Toxicity】SR-MMP
OTHER FACTORS ABOUT TRANSFOMATION:
Credibility
:
None
None
Qualified
High
Variance
:
None
None
No Change
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